TRP Channel Inhibitors

TRPC

TRPM

TRPV

TRPA

TRPML

TRP Channel Inhibitors, Agonists, Antagonists, Activators & Modulators

Product Name	TRPC	TRPM	TRPV	TRPA	TRPML	Purity
Rosiglitazone	TRPC5, EC₅₀: 30 μM					99.94%
Anandamide			TRPV1			≥99.0%
SOR-C13 acetate			TRPV6, IC₅₀: 14 nM			98.56%
GSK1016790A			TRPV4			99.79%
ML-SI3					TRPML1, IC₅₀: 4.7 μM	99.93%
SB-366791			hTRPV1, IC₅₀: 5.7 nM			98.11%
GSK1702934A	TRPC3					≥99.0%
Icilin		TRPM8				99.26%
Dihydrocapsaicin			TRPV1			99.86%
ML204	TRPC4 TRPC5					99.08%
CIM0216		TRPM3				99.94%
(1R,2R)-ML-SI3					TRPML1, IC₅₀: 1.6 μM TRPML2, IC₅₀: 2.3 μM TRPML3, IC₅₀: 12.5 μM	99.45%
JNJ-28583113		TRPM2				98.06%
Pyr10	TRPC3, IC₅₀: 0.72 μM					99.42%
Acoltremon		TRPM8				99.90%
SET2			TRPV2, IC₅₀: 0.46 μM			99.72%
Englerin A	hTRPC4, EC₅₀: 11.2 nM hTRPC5, EC₅₀: 7.6 nM					99.50%
(rel)-ML-SI3					TRPML1, IC₅₀: 3.1 μM TRPML2, EC₅₀: 3.3 μM TRPML3, IC₅₀: 28.5 μM	99.81%
LE135			TRPV1, EC₅₀: 2.5 μM	TRPA1, EC₅₀: 20 μM		99.03%
SOR-C13 TFA			TRPV6, IC₅₀: 14 nM			99.18%
Rosiglitazone hydrochloride	TRPC5, EC₅₀: 30 μM					99.31%
AP-18				TRPA1, IC₅₀: ~3 μM		99.80%
RQ-00203078		TRPM8, IC₅₀: 5.3 nM (Rat TRPM8 channels) TRPM8, IC₅₀: 8.3 nM (Human TRPM8 channels)	TRPV4, IC₅₀: 10 μM			99.84%
TRPV2-selective blocker 1			TRPV2, IC₅₀: 6.3 μM			99.84%
PF-04745637				TRPA1, IC₅₀: 17 nM		99.97%
Larixyl acetate	hTRPC6, IC₅₀: 0.58 μM hTRPC3, IC₅₀: 6.83 μM					99.46%
Ononetin		TRPM3, IC₅₀: 0.3 μM				99.54%
JNJ-17203212			TRPV1			99.94%
Capsiate			TRPV1			99.51%
TRPV3 antagonist 74a			TRPV3			99.85%
M8-B		TRPM8				99.89%
ML204 hydrochloride	TRPC4 TRPC5					99.70%
Phenamil methanesulfonate	TRPC3, IC₅₀: 140 nM					≥98.0%
MSP-3			TRPV1, EC₅₀: 0.87 μM			98.53%
Chembridge-5861528				TRPA1, IC₅₀: 14.3 μM (allyl isothiocyanate-evoked TRPA1 response) TRPA1, IC₅₀: 18.7 μM (4-HNE-evoked TRPA1 response)		99.76%
TRPV1 antagonist 3		TRPM8, IC₅₀: 7.45 μM	hTRPV1, IC₅₀: 2.66 nM			99.30%
(1S,2S)-ML-SI3					TRPML1, IC₅₀: 5.9 μM TRPML2, EC₅₀: 2.7 μM TRPML3, EC₅₀: 10.8 μM	99.82%
AS1269574				TRPA1		99.84%
MDR-652			hTRPV1, Ki: 11.4 nM rTRPV1, Ki: 23.8 nM hTRPV1, EC₅₀: 5.05 nM rTRPV1, EC₅₀: 93 nM			99.02%
TRPA1-IN-2				TRPA1, IC₅₀: 0.04 μM		99.82%
Vanilloid receptor antagonist 1			TRPV1			99.54%
Olvanil			TRPV1, EC₅₀: 0.7 nM			≥99.0%
Chrysin 6-C-glucoside 8-C-arabinoside			TRPV1			99.11%
17(R)-Resolvin D1			TRPV3, IC₅₀: 398 nM			99.1%
D-erythro-Sphingosine hydrochloride		TRPM3
ABT-102			TRPV1
SOR-C13			TRPV6, IC₅₀: 14 nM			98.56%
RN-1665			hTRPV4, IC₅₀: 0.26 μM rTRPV4, IC₅₀: 0.39 μM			99.93%
FAAH/TRPV1 blocker-1			TRPV1, IC₅₀: 94.9 μM
Methyl kakuol				TRPA1
TRPV4 antagonist 4			TRPV4, IC₅₀: 22.65 nM
JTS-653			TRPV1
TRPC antagonist 1	TRPC3, IC₅₀: 2.4 μM TRPC4, IC₅₀: 12.2 μM TRPC5, IC₅₀: 7.6 μM TRPC6, IC₅₀: 2.9 μM TRPC7, IC₅₀: 3.4 μM
JW-65	TRPC3
TRPV4-IN-5			TRPV4, IC₅₀: 0.46 μM
TRPV1-IN-2				TRPA1
L-R4W2 TFA			TRPV1, IC₅₀: 0.1 μM
(R)-Methanandamide			TRPV1
L687	TRPC3 TRPC6 TRPC7
TRPC4/5-IN-1	TRPC5, IC₅₀: 0.54 μM TRPC4, IC₅₀: 2.06 μM
TRPC4/5-IN-2	TRPC5
5-Iodoresiniferatoxin			rTRPV1, IC₅₀: 0.7 nM hTRPV1, IC₅₀: 5.4 nM
L-R4W2			TRPV1, IC₅₀: 0.1 μM
MK-2295			TRPV1
GDC-0334				TRPA1
Xeniafaraunol A		TRPM7
Dihydrocapsiate			TRPV1			99.18%
TRPV1/CB2 agonist 1			TRPV1, EC₅₀: 26.8 μM
TRPV1 antagonist 5			TRPV1
AMG8788				TRPA1, IC₅₀: 1 μM
AMG9678				TRPA1, IC₅₀: 0.6 μM
Scalaradial		TRPM2, IC₅₀: 210 nM TRPM7, IC₅₀: 760 nM
N-Arachidonyldopamine			TRPV1, EC₅₀: ~50 nM			98.36%
TRPM8-IN-1		TRPM8, IC₅₀: <5 μM
TRPC5-IN-4	TRPC5, IC₅₀: 14.07 nM TRPC4, IC₅₀: 65 nM
V116517			TRPV1
Protokylol hydrochloride			TRPV1
N-Arachidonoyl Taurine			TRPV1, EC₅₀: 28 μM TRPV4, Ki: 21 μM
TRPV6-IN-1			TRPV6
TRPA1-IN-3				TRPA1

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